API Intermediates

Structure Name of Compound Name of
Intermediates
CAS NO
4,6-DICHLORO-2-(PROPYLTHIO)PYRIMIDIN-5-AMINE TICAGRELOR [145783-15-9]
(1R,2S)-2-(3,4-DIFLUOROPHENYL)CYCLOPROPANAMINIUM (2R)-HYDROXY(PHENYL)ETHANOATE TICAGRELOR [376608-71-8]
2-(((3AR,4S,6R,6AS)-6-AMINO-2,2-DIMETHYLTETRAHYDRO-3AH-CYCLOPENTA[D][1,3]DIOXOL-4-YL)OXY)ETHANOL (2R,3R)-2,3-DIHYDROXYSUCCINATE TICAGRELOR [376608-65-0]
3-(((3aR,4S,6R,6aS)-6-((5-amino-6-chloro-2-(propylthio)pyrimidin-4-yl)amino)-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4-yl)oxy)propan-1-ol TICAGRELOR [376608-74-1]
ETHANOL, 2-[[(3AR,4S,6R,6AS)-6-[7-CHLORO-5-(PROPYLTHIO)-3H-1,2,3-TRIAZOLO[4,5-D]PYRIMIDIN-3-YL]TETRAHYDRO-2,2-DIMETHYL-4H-CYCLOPENTA-1,3-DIOXOL-4-YL]OXY]- TICAGRELOR [376608-75-2]
2-(((3aR,4S,6R,6aS)-6-(7-(((1R,2S)-2-(3,4-ifluorophenyl)cyclopropyl)amino)-5-(propylthio)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)-2,2-dimethyltetrahydro-4H-cyclopenta[d][1,3]dioxol-4-yl)oxy)ethan-1-ol TICAGRELOR [274693-26-4]
(1S,2S,3R,5S)-3-(7-(((1R,2S)-2-(3,4-difluorophenyl)cyclopropyl)amino)-5-(propylthio)- 3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)-5-(2-hydroxyethoxy)cyclopentane-1,2-diol TICAGRELOR [274693-27-5]
(6aR,9R)-7-allyl-4,6,6a,7,8,9,10,10a-octahydroindolo[4,3-fg]quinoline-9-carboxylic acid TICAGRELOR [81409-74-7]
ALPHA-ERGOCRYPTINE TICAGRELOR [511-09-1]
(3S,8aS)-3-isobutylhexahydropyrrolo[1,2-a]pyrazine-1,4-dione TICAGRELOR [2873-36-1]
(6aR,9R,10aR)-7-allyl-N-(3-(dimethylamino)propyl)-N-(ethylcarbamoyl)- 4,6,6a,7,8,9,10,10a-octahydroindolo[4,3-fg]quinoline-9-carboxamide TICAGRELOR [81409-90-7]
4,5-dimethyl 1,3-dioxolen Olmesatan intermediates [37830-90-3]
2-Propyl-1H-imidazole-4,5-dicarboxylic acid dimethyl ester Structure 2-propyl Imidazole 4,5 bicarboxylic Acid diethyl Ester Olmesatan intermediates [124750-59-0]
9-Benzyloxy-3-(2-Chloroethyl)-2-methyl pyrido
[1,2-a]pyrimidine-4-one
Paliperidone intermediate [147687-17-0]
4-chloro-6-ethyl-5-fluoropyrimidine voriconazole intermediate [137234-74-3]
Methyl(3R)-3-(tert-butyldimethylsilyloxy)-5-oxo-6-triphenylphosphoranylidenehexanoate Rosuvastatin intermediate [154026-95-6]
2-oxo-2,4,5,6,7,7a-hexahydrothieno [3,2-c] pyridine
Hydrocloride
Prasugrel Intermediate [115473-15-9]
1-(Mercaptomethyl)cyclopropane]acetic acid Montelukast intermediates [162515-68-6]
2-[1-( Hydroxymethyl)-cyclopropane]-acetonitrile Montelukast intermediates [152922-71-9]
Meldrum's acid Montelukast intermediates [2033-24-1]
BOC-D-SERINE Lacosamide intermediates [6368-20-3]
(R)-tert-Butyl 1-(benzylamino)-3-methoxy-1-
oxopropan-2-ylcarbamate
Lacosamide Intermediate [880468-89-3]
(4-Fluorobenzoyl)butyric acid Ezetimibe intermediates [149437-76-3]
(4S)-3-[5-(4-Fluorophenyl)-1,5-dioxopenyl]-4-
phenyl-2-oxazolidinone
Ezetimibe [189028-93-1]
4-[(4-Fluorophenyl)imino]methyl]-phenol Ezetimibe [3382-63 ]
(S)-3-(aminomethyl)-5-methylhexanoic acid Pragabalin [148553-50-8]
3-[(3-Amino-4-methylaminobenzoyl)pyridin-2-
ylamino]propionic acid ethyl ester
DABIGATRAN [212322-56-0]
3-[2-(4-Cyanophenyl)amino]methyl]-1-methyl-1H-
benzimidazol-5-yl] carbonyl]pyridin-2-ylamino]
propionic acid ethyl ester.
DABIGATRAN [211915-84-3]
3-ethyl-5-methyl-2-[(2-phthalamidoethoxy) methyl]

-4-(2-chlorophenyl)-1, 4-dihydro-6-methyl

-3,5-pyridinedicarboxylate

Amlodipine Besylate [88150-62-3]
2-[(2-aminoethoxy)methyl]-4-(2-chlorophenyl)
-1,4-dihydro-6-methyl-3,5-pyridine dicarboxylic acid
-3-ethyl-5-methyl ester

Amlodipine Besylate [88150-42-9]
(+)-2-(2-chlorophenyl)-N-(2-thienyl) ethyl)

Glycine methyl ester hydrochloride

Clopidogrel Bisulfate [88150-62-3]
Thieno (3, 2-C)-4,5,6,7-tetra hydro pyridine
hydrochloride
Clopidogrel Bisulfate [28783-41-7]
2-amino-5-methyl thiophene-3-carbonitrile Olanzapine [138564-58-6]
2-(2-Nitro anilino)-5-methyl thiophene-3-
carbonitrile
Olanzapine [138564-59-7]
4-amino-2-methyl-10H-thieno [2,3-b][1,5]
benzodiazepine
hydrochloride

Olanzapine [138564-60-0]
2-methyl-4-(4-methyl-1-piperazinyl)- 10H-thieno

[2,3-b][1,5]benzodiazepine

Olanzapine [132539-06-1]
2-(4-methyl-2-phenyl piperazin-1-yl)
pyridine-3-carboxylic acid
Mirtazapine Mol. F: C17H19N3 O2
1-(3-Hydroxymethylpyridin-2-yl)-4-methyl-2-
phenylpiperazine
Mirtazapine [61337-89-1]
1-Benzylpiperidine-4-carbaldehyde Donepezil [22065-85-6]
2-(1-Benzylpiperidin-4-ylmethylene)-5,
6-dimethoxy indan-1-one
DONEPEZIL [142057-77-0]
N-[(2'-Cyano-(1,1'-biphenyl)-4-yl)methyl)]valine
methyl ester hydrochloride

Valsartan CAS # [137863-89-9]
(S)-Methyl 2-(N-((2'-cyanobiphenyl-4-yl)methyl)

pentanamido) -3-methylbutanoate

Valsartan [137863-90-2]
N-[(2’-Cyanobiphenyl-4-yl) methyl]-L-
valine benzyl ester
Valsartan [137864-23-4]
2,3:4,5-Bis - O-(1-Methyl Ethylidene)-Β-
Fructopyranose
Topiramate [20880-92-6]
2,3:4,5-Bis-O-(1-methylethylidene)-beta –D-
fructopyranose sulfate
TOPIRAMATE [97240-79-4]
S-N-[[3-[3-Fluoro-4-[4-morpholinyl]phenyl]
-2-oxo-5-oxazolidinyl]methyl]amine
Linezolid Mol.F: C14H18FN3O3
4-BROMOMETHYL-[2'-(2- TRITYL-2H-TETRAZOL-
5-YL)] BIPHENYL
Losartan
Condesartan Olmesartan
Irbesartan
[133051-88-4]
8-chloro-5,6-dihydro-11H-benzo[5,6]cyclohepta
[1,2-b]pyridin-11-one
LORATADINE [31251-41-9]
3-[2-(3-Chlorophenyl)ethyl]-2-pyridine carbonitrile LORATADINE [31255-57-9]
9-(4-ACETOXY-3-ACETOXYMETHYLBUTYL)-2-
AMINO-6-CHLOROPURINE
FAMCYCLOVIR [1020718-81-3]
4-Hydroxy benzothioamide FEBUXOSTAT [25984-63-8]
Ethyl 2-(4-hydroxyphenyl)-4-methylthiazole-5-carboxylate FEBUXOSTAT [161797-99-5]
Ethyl 2-(3-formyl-4-hydroxyphenyl)-4-methyl thiazole-5-
carboxylate
FEBUXOSTAT [ 161798-01-2]
Ethyl-2-(3-formyl-4-isobutoxyphenyl)-4-
methylthiazole-5-carboxylate
FEBUXOSTAT [161798-03-4]
Ethyl-2-(3-Cyano-4-isobutoxyphenyl)-4-
methyl-5-thiocarboxylate
FEBUXOSTAT [160844-75-7]
(3R)-3-(2-AMINO-2-OXOETHYL)-5-
METHYLHEXANOIC ACID
PREGABALIN [181289-33-8]
6-Methoxy-2-(4-methoxyphenyl)benzobithiophene RALOXIFINE [181289-33-8]
4-[2-(1-Pipiridine) ethoxybenzoic acid hydrochloride RALOXIFINE [84449-80-9]
ethyl 4-[(4-chloro-2-nitrophenyl)amino]piperidine-1-
carboxylate
DOMPERIDONE [53786-44-0]
5-chloro-1-(piperidin-4-yl)-1,3-dihydro-2H-
benzimidazol-2-one
DOMPERIDONE [53786-28-0]
1-(3-Chloropropyl)-1,3-dihydro-2H-
benzimidazol-2-one
DOMPERIDONE [62780-89-6]
5-(phenylcarbonyl)-2,3-dihydro-1H-
pyrrolizine-1-carboxylic acid
KETOROLAC [74103-06-3]
Benzeneaceticacid, 4-[4-[4-(hydroxydiphenylmethyl)-1
piperidinyl] -1-oxobutyl]-a,a-dimethyl-, methyl ester

FEXOFENADINE [154477-55-1]